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The Sign of Nuclear Magnetic Resonance Chemical Shift Difference as a Determinant of the Origin of Binding Selectivity: Elucidation of the Position Dependence of Phosphorylation in Ligands Binding to Scribble PDZ1.

Biochemistry. 2018 Jan 09;57(1):66-71. doi:10.1021/acs.biochem.7b00965. Epub 2017 Nov 27
Gustav N Sundell 1 , Beat Vögeli 2 , Ylva Ivarsson 1 , Celestine N Chi 3
Gustav N Sundell 1 , Beat Vögeli 2 , Ylva Ivarsson 1 , Celestine N Chi 3

[No authors listed]

Author information
  • 1 Department of Chemistry, Uppsala University , BMC Box 576, SE-75123 Uppsala, Sweden.
  • 2 Department of Biochemistry and Molecular Genetics, University of Colorado at Denver , 12801 East 17th Avenue, Aurora, Colorado 80045, United States.
  • 3 Department of Medical Biochemistry and Microbiology, Uppsala University , BMC Box 582, SE-75123 Uppsala, Sweden.

摘要


H shift changes of the PDZ1 domain of Scribble upon interaction with two pairs of phosphorylated and unphosphorylated peptides. We find that detailed differences in the molecular basis of this PDZ-ligand interaction can be obtained from our analysis to which the classical method of combined chemical shift perturbation analysis is insensitive. In addition, we find a correlation between affinity and millisecond motions. Application of the methodology to Cyclophilin a, a cis-trans isomerase, reveals molecular details of peptide recognition. We consider our directionality vector chemical shift analysis as a method of choice when distinguishing the molecular origin of binding specificities of a class of similar ligands, which is often done in drug discovery.